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Silidianin

PubChem CID: 11982272

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Compound Synonyms Silydianin, 29782-68-1, Silidianin, Silidianine, Silidianina, Silidianin [INN], Silidianinum, Silidianine [INN-French], Silidianinum [INN-Latin], Silidianina [INN-Spanish], UNII-7P89L7W179, EINECS 249-848-5, SILIDIANIN [MART.], SILYDIANIN [USP-RS], DTXSID70858696, 7P89L7W179, Silidianine (INN-French), Silidianinum (INN-Latin), Silidianina (INN-Spanish), SILIDIANIN (MART.), SILYDIANIN (USP-RS), (1R,3R,6R,7R,10R)-3-hydroxy-10-(4-hydroxy-3-methoxyphenyl)-8-[(2R,3R)-3,5,7-trihydroxy-4-oxo-2,3-dihydrochromen-2-yl]-4-oxatricyclo[4.3.1.03,7]dec-8-en-2-one, (1S,3S,6R,7S,10R)-3-Hydroxy-10-(4-hydroxy-3-methoxyphenyl)-8-[(2R,3R)-3,5,7-trihydroxy-4-oxo-2,3-dihydrochromen-2-yl]-4-oxatricyclo[4.3.1.03,7]dec-8-en-2-one, SILIDIANIN (CONSTITUENT OF MILK THISTLE) [DSC], (+)-2,3.ALPHA.,3A.ALPHA.A,7A-TETRAHYDRO-7A.ALPHA.-HYDROXY-8-(4-HYDROXY-3-METHOXYPHENYL)-4-(3.ALPHA.,5,7-TRIHYDROXY-4-OXO-2.BETA.-CHROMANYL)-3,6-METHANOBENZOFURAN-7(6.ALPHA.H)-ONE, Silydianin (Standard), Silydianin, analytical standard, CHEMBL2397733, HY-N0646R, DTXCID20809436, CYGIJEJDYJOUAN-JSGXPVSSSA-N, HY-N0646, AKOS030573534, FS42773, (+)-2,3 alpha,3a alpha,7a-tetrahydro-7aalpha-hydroxy-8-(4-hydroxy-3-methoxyphenyl)-4-(3alpha,5,7-trihydroxy-4-oxo-2beta-chromanyl)-3,6-methanobenzofuran-7(6alphaH)-one, AC-34761, AS-56229, CS-0009672, SILIDIANIN (CONSTITUENT OF MILK THISTLE), BRD-K52002287-001-01-0, Q27268678, Silydianin, United States Pharmacopeia (USP) Reference Standard, (+)-2,3alpha,3aalpha,7a-Tetrahydro-7aalpha-hydroxy-8-(4-hydroxy-3-methoxyphenyl)-4-(3alpha,5,7-trihydroxy-4-oxo-2beta-chromanyl)-3,6-methanobenzofuran-7(6alphaH)-one, (+)-2,3ALPHA,3AALPHAA,7A-TETRAHYDRO-7AALPHA-HYDROXY-8-(4-HYDROXY-3-METHOXYPHENYL)-4-(3ALPHA,5,7-TRIHYDROXY-4-OXO-2BETA-CHROMANYL)-3,6-METHANOBENZOFURAN-7(6ALPHAH)-ONE, (3R,3aR,6R,7aR,8R)-7a-Hydroxy-8-(4-hydroxy-3-methoxyphenyl)-4-((2R,3R)-3,5,7-trihydroxy-4-oxochroman-2-yl)-3,3a,6,7a-tetrahydro-3,6-methanobenzofuran-7(2H)-one, 249-848-5
Ghose Rule False
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 163.0
Hydrogen Bond Donor Count 5.0
Pfizer 3 75 Rule True
Scaffold Graph Level CC1CC(C2CC3C(C)C4CCC(C3C3CCCCC3)C24)CC2CCCCC12
Np Classifier Class Dihydroflavonols, Flavonolignans
Deep Smiles COcccccc6O))))[C@@H][C@H]CO[C@@][C@H]5C=C[C@H]9C6=O))))[C@H]OcccO)ccc6C=O)[C@@H]%10O))))O))))))))))O
Heavy Atom Count 35.0
Classyfire Class Flavonoids
Scaffold Graph Node Level OC1CC(C2CC3C(O)C4OCC(C3C3CCCCC3)C24)OC2CCCCC12
Classyfire Subclass Flavans
Isotope Atom Count 0.0
Molecular Complexity 935.0
Database Name cmaup_ingredients;imppat_phytochem;npass_chem_all;pubchem
Defined Atom Stereocenter Count 7.0
Uniprot Id n.a., O42713
Iupac Name (1R,3R,6R,7R,10R)-3-hydroxy-10-(4-hydroxy-3-methoxyphenyl)-8-[(2R,3R)-3,5,7-trihydroxy-4-oxo-2,3-dihydrochromen-2-yl]-4-oxatricyclo[4.3.1.03,7]dec-8-en-2-one
Prediction Hob 0.0
Veber Rule False
Classyfire Superclass Phenylpropanoids and polyketides
Xlogp 0.8
Gsk 4 400 Rule False
Molecular Formula C25H22O10
Scaffold Graph Node Bond Level O=C1CC(C2=CC3C(=O)C4OCC(C24)C3c2ccccc2)Oc2ccccc21
Prediction Swissadme 0.0
Inchi Key CYGIJEJDYJOUAN-JSGXPVSSSA-N
Silicos It Class Soluble
Fcsp3 0.36
Logs -3.521
Rotatable Bond Count 3.0
Logd 1.717
Synonyms silydianin
Esol Class Soluble
Functional Groups CC=C(C)C, CO, CO[C@@](C)(O)C(C)=O, cC(C)=O, cO, cOC
Compound Name Silidianin
Prediction Hob Swissadme 0.0
Exact Mass 482.121
Formal Charge 0.0
Monoisotopic Mass 482.121
Hydrogen Bond Acceptor Count 10.0
Molecular Weight 482.4
Gi Absorption False
Covalent Unit Count 1.0
Total Atom Stereocenter Count 7.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 True
Esol -3.3908484857142867
Inchi InChI=1S/C25H22O10/c1-33-16-4-9(2-3-14(16)27)18-11-7-12(20-13(18)8-34-25(20,32)24(11)31)23-22(30)21(29)19-15(28)5-10(26)6-17(19)35-23/h2-7,11,13,18,20,22-23,26-28,30,32H,8H2,1H3/t11-,13-,18+,20+,22+,23-,25-/m1/s1
Smiles COC1=C(C=CC(=C1)[C@@H]2[C@H]3CO[C@@]4([C@H]3C(=C[C@H]2C4=O)[C@@H]5[C@H](C(=O)C6=C(C=C(C=C6O5)O)O)O)O)O
Nring 7.0
Np Classifier Biosynthetic Pathway Shikimates and Phenylpropanoids
Defined Bond Stereocenter Count 0.0
Egan Rule False
Np Classifier Superclass Lignans, Flavonoids

  • 1. Outgoing r'ship FOUND_IN to/from Silybum Marianum (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all