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Galanthamine N-Oxide

PubChem CID: 11748698

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Compound Synonyms Galanthamine N-Oxide, Galantamine N-Oxide, 134332-50-6, 199014-26-1, UNII-S6AF61T5WO, S6AF61T5WO, (1S,12S,14R)-9-methoxy-4-methyl-4-oxido-11-oxa-4-azoniatetracyclo[8.6.1.01,12.06,17]heptadeca-6(17),7,9,15-tetraen-14-ol, DTXSID40173681, GALANTAMINE METABOLITE M10, GALANTHAMINE (RS)-N-OXIDE, Galanthamine-N-oxide, (4AS-(4A.ALPHA.,6.BETA.,8AR*))-4A,5,9,10,11,12-HEXAHYDRO-3-METHOXY-11-METHYL-6H-BENZOFURO(3A,3,2-EF)(2)BENZAZEPIN-6-OL, N-OXIDE, 6H-BENZOFURO(3A,3,2-EF)(2)BENZAZEPIN-6-OL, 4A,5,9,10,11,12-HEXAHYDRO-3-METHOXY-11-METHYL-, 11-OXIDE, (4AS,6R,8AS)-, 6H-BENZOFURO(3A,3,2-EF)(2)BENZAZEPIN-6-OL, 4A,5,9,10,11,12-HEXAHYDRO-3-METHOXY-11-METHYL-, 11-OXIDE, (4AS-(4A.ALPHA.,6.BETA.,8AR*))-, (1S,12S,14R)-9-methoxy-4-methyl-4-oxido-11-oxa-4-azoniatetracyclo(8.6.1.01,12.06,17)heptadeca-6(17),7,9,15-tetraen-14-ol, (4aS,6R,8aS)-4a,5,9,10,11,12-Hexahydro-3-methoxy-11-methyl-6H-benzofuro[3a,3,2-ef][2]benzazepin-6-ol 11-oxide, SCHEMBL3299153, DTXCID2096172, LROQBKNDGTWXET-FVWDGWMTSA-N, AKOS030241457, FG23640, GALANTAMINE N-OXIDE [USP IMPURITY], DB-257732, Galanthamine 10-Oxide(Galanthamine N-Oxide), NS00116587, Q27288725, GALANTAMINE HYDROBROMIDE IMPURITY, 6.BETA.-HEXAHYDROGALANTAMINE-[USP IMPURITY], GALANTAMINE HYDROBROMIDE IMPURITY, 6BETA-HEXAHYDROGALANTAMINE-(USP IMPURITY), (4As,6r,8as)-3-methoxy-11-methyl-5,6,9,10,11,12-hexahydro-4aH-[1]benzofuro[3a,3,2-ef][2]benzazepin-6-ol 11-oxide, (4aS,6R,8aS)-4a,5,9,10,11,12-Hexahydro-3-methoxy-11-methyl-6H-benzofuro[3a,3,2-ef][2]benzazepin-6-ol 11-oxide, 6H-Benzofuro[3a,3,2-ef][2]benzazepin-6-ol, 4a,5,9,10,11,12-hexahydro-3-methoxy-11-methyl-, 11-oxide, (4aS,6R,8aS)-, 6H-Benzofuro[3a,3,2-ef][2]benzazepin-6-ol, 4a,5,9,10,11,12-hexahydro-3-methoxy-11-methyl-, 11-oxide, [4aS-(4aa,6ss,8aR*)]-, (4aS,6R,8aS,11R)-4a,5,9,10,11,12-Hexahydro-3-methoxy-11-methyl-6H-benzofuro[3a,3,2-ef][2]benzazepin-6-ol 11-oxide, Nivalin-oxide, Gala nthamine 10-oxide, (4AS-(4AALPHA,6BETA,8AR*))-4A,5,9,10,11,12-HEXAHYDRO-3-METHOXY-11-METHYL-6H-BENZOFURO(3A,3,2-EF)(2)BENZAZEPIN-6-OL, N-OXIDE, 6H-BENZOFURO(3A,3,2-EF)(2)BENZAZEPIN-6-OL, 4A,5,9,10,11,12-HEXAHYDRO-3-METHOXY-11-METHYL-, 11-OXIDE, (4AS-(4AALPHA,6BETA,8AR*))-
Ghose Rule True
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 56.8
Hydrogen Bond Donor Count 1.0
Pfizer 3 75 Rule False
Scaffold Graph Level C1CCC23CCCCC2CC2CCCC(C1)C23
Np Classifier Class Amarylidaceae alkaloids
Deep Smiles COcccccc6O[C@@H][C@]5C=C[C@@H]C6)O))))CC[N+]C%10)[O-])C
Heavy Atom Count 22.0
Classyfire Class Amaryllidaceae alkaloids
Scaffold Graph Node Level C1CC2CNCCC34CCCCC3OC(C1)C24
Classyfire Subclass Galanthamine-type amaryllidaceae alkaloids
Isotope Atom Count 0.0
Molecular Complexity 483.0
Database Name imppat_phytochem;pubchem
Defined Atom Stereocenter Count 3.0
Iupac Name (1S,12S,14R)-9-methoxy-4-methyl-4-oxido-11-oxa-4-azoniatetracyclo[8.6.1.01,12.06,17]heptadeca-6(17),7,9,15-tetraen-14-ol
Veber Rule True
Classyfire Superclass Alkaloids and derivatives
Xlogp 1.3
Gsk 4 400 Rule True
Molecular Formula C17H21NO4
Scaffold Graph Node Bond Level C1=CC23CC[NH2+]Cc4cccc(c42)OC3CC1
Inchi Key LROQBKNDGTWXET-FVWDGWMTSA-N
Silicos It Class Soluble
Rotatable Bond Count 1.0
Synonyms galanthamine n-oxide
Esol Class Soluble
Functional Groups CC=CC, CO, C[N+](C)(C)[O-], cOC
Compound Name Galanthamine N-Oxide
Exact Mass 303.147
Formal Charge 0.0
Monoisotopic Mass 303.147
Hydrogen Bond Acceptor Count 4.0
Molecular Weight 303.35
Gi Absorption True
Covalent Unit Count 1.0
Total Atom Stereocenter Count 4.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 True
Inchi InChI=1S/C17H21NO4/c1-18(20)8-7-17-6-5-12(19)9-14(17)22-16-13(21-2)4-3-11(10-18)15(16)17/h3-6,12,14,19H,7-10H2,1-2H3/t12-,14-,17-,18?/m0/s1
Smiles C[N+]1(CC[C@@]23C=C[C@@H](C[C@@H]2OC4=C(C=CC(=C34)C1)OC)O)[O-]
Np Classifier Biosynthetic Pathway Alkaloids
Defined Bond Stereocenter Count 0.0
Egan Rule True
Np Classifier Superclass Tyrosine alkaloids

  • 1. Outgoing r'ship FOUND_IN to/from Lycoris Radiata (Plant) Rel Props:Reference:ISBN:9788185042145