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Chiapenine ES-I

PubChem CID: 11182206

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Compound Synonyms Chiapenine ES-I, ((1S,3R,18S,19R,20R,21R,22S,23R,24R,25R,26S)-22,23,25-triacetyloxy-21-(acetyloxymethyl)-20-benzoyloxy-15,26-dihydroxy-3,15,26-trimethyl-6,16-dioxo-2,5,17-trioxa-11-azapentacyclo(16.7.1.01,21.03,24.07,12)hexacosa-7(12),8,10-trien-19-yl) benzoate, (1R,3R,15S,18S,19S,20S,21S,22R,23R,24S,25R,26S)-22,23,25-Tris(acetyloxy)-21-((acetyloxy)methyl)-20-(benzoyloxy)-15,26-dihydroxy-3,15,26-trimethyl-6,16-dioxo-2,5,17-trioxa-11-azapentacyclo(16.7.1.0,.0,.0,)hexacosa-7(12),8,10-trien-19-yl benzoic acid, (1R,3R,15S,18S,19S,20S,21S,22R,23R,24S,25R,26S)-22,23,25-Tris(acetyloxy)-21-[(acetyloxy)methyl]-20-(benzoyloxy)-15,26-dihydroxy-3,15,26-trimethyl-6,16-dioxo-2,5,17-trioxa-11-azapentacyclo[16.7.1.0,.0,.0,]hexacosa-7(12),8,10-trien-19-yl benzoic acid, [(1S,3R,18S,19R,20R,21R,22S,23R,24R,25R,26S)-22,23,25-triacetyloxy-21-(acetyloxymethyl)-20-benzoyloxy-15,26-dihydroxy-3,15,26-trimethyl-6,16-dioxo-2,5,17-trioxa-11-azapentacyclo[16.7.1.01,21.03,24.07,12]hexacosa-7(12),8,10-trien-19-yl] benzoate, CHEMBL505015, 654670-28-7
Topological Polar Surface Area 273.0
Hydrogen Bond Donor Count 2.0
Heavy Atom Count 68.0
Isotope Atom Count 0.0
Molecular Complexity 1980.0
Database Name cmaup_ingredients;pubchem
Defined Atom Stereocenter Count 11.0
Iupac Name [(1S,3R,18S,19R,20R,21R,22S,23R,24R,25R,26S)-22,23,25-triacetyloxy-21-(acetyloxymethyl)-20-benzoyloxy-15,26-dihydroxy-3,15,26-trimethyl-6,16-dioxo-2,5,17-trioxa-11-azapentacyclo[16.7.1.01,21.03,24.07,12]hexacosa-7(12),8,10-trien-19-yl] benzoate
Prediction Hob 0.0
Xlogp 2.9
Molecular Formula C48H51NO19
Prediction Swissadme 0.0
Inchi Key QIADRFASJTYLCV-CSQIADDDSA-N
Fcsp3 0.4791666666666667
Logs -3.572
Rotatable Bond Count 15.0
Logd 1.504
Compound Name Chiapenine ES-I
Prediction Hob Swissadme 0.0
Exact Mass 945.306
Formal Charge 0.0
Monoisotopic Mass 945.306
Hydrogen Bond Acceptor Count 20.0
Molecular Weight 945.9
Covalent Unit Count 1.0
Total Atom Stereocenter Count 12.0
Total Bond Stereocenter Count 0.0
Esol -6.737611152941176
Inchi InChI=1S/C48H51NO19/c1-25(50)60-24-47-38(64-28(4)53)34(62-26(2)51)33-36(63-27(3)52)48(47)46(7,59)37(35(65-40(54)29-15-10-8-11-16-29)39(47)66-41(55)30-17-12-9-13-18-30)67-43(57)44(5,58)21-20-32-31(19-14-22-49-32)42(56)61-23-45(33,6)68-48/h8-19,22,33-39,58-59H,20-21,23-24H2,1-7H3/t33-,34-,35+,36-,37+,38-,39+,44?,45+,46+,47-,48+/m1/s1
Smiles CC(=O)OC[C@]12[C@@H]([C@@H]([C@@H]3[C@H]([C@]14[C@@]([C@H]([C@@H]([C@@H]2OC(=O)C5=CC=CC=C5)OC(=O)C6=CC=CC=C6)OC(=O)C(CCC7=C(C=CC=N7)C(=O)OC[C@@]3(O4)C)(C)O)(C)O)OC(=O)C)OC(=O)C)OC(=O)C
Nring 7.0
Defined Bond Stereocenter Count 0.0

  • 1. Outgoing r'ship FOUND_IN to/from Maytenus Chiapensis (Plant) Rel Props:Source_db:cmaup_ingredients