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2'',3''-Dihydrocephalomannine

PubChem CID: 10509711

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Compound Synonyms Dihydrocephalomannin?e, Dihydrocephalomannine, 159001-25-9, 2'',3''-Dihydrocephalomannine, N-Debenzoyl-N-a-methylbutyrylpaclitaxel, OKEKLOJNCOIPIT-DYMXBOOHSA-, [(1S,2S,3R,4S,7R,9S,10S,12R,15S)-4,12-diacetyloxy-1,9-dihydroxy-15-[(2R,3S)-2-hydroxy-3-(2-methylbutanoylamino)-3-phenylpropanoyl]oxy-10,14,17,17-tetramethyl-11-oxo-6-oxatetracyclo[11.3.1.03,10.04,7]heptadec-13-en-2-yl] benzoate, InChI=1/C45H55NO14/c1-9-23(2)39(52)46-33(27-16-12-10-13-17-27)34(50)41(54)58-29-21-45(55)38(59-40(53)28-18-14-11-15-19-28)36-43(8,30(49)20-31-44(36,22-56-31)60-26(5)48)37(51)35(57-25(4)47)32(24(29)3)42(45,6)7/h10-19,23,29-31,33-36,38,49-50,55H,9,20-22H2,1
Topological Polar Surface Area 221.0
Hydrogen Bond Donor Count 4.0
Heavy Atom Count 60.0
Isotope Atom Count 0.0
Molecular Complexity 1730.0
Database Name cmaup_ingredients;pubchem
Defined Atom Stereocenter Count 11.0
Iupac Name [(1S,2S,3R,4S,7R,9S,10S,12R,15S)-4,12-diacetyloxy-1,9-dihydroxy-15-[(2R,3S)-2-hydroxy-3-(2-methylbutanoylamino)-3-phenylpropanoyl]oxy-10,14,17,17-tetramethyl-11-oxo-6-oxatetracyclo[11.3.1.03,10.04,7]heptadec-13-en-2-yl] benzoate
Prediction Hob 0.0
Xlogp 2.2
Molecular Formula C45H55NO14
Prediction Swissadme 0.0
Inchi Key OKEKLOJNCOIPIT-DYMXBOOHSA-N
Fcsp3 0.5555555555555556
Logs -3.774
Rotatable Bond Count 15.0
Logd 1.636
Compound Name 2'',3''-Dihydrocephalomannine, N-Debenzoyl-N-a-methylbutyrylpaclitaxel
Prediction Hob Swissadme 0.0
Exact Mass 833.362
Formal Charge 0.0
Monoisotopic Mass 833.362
Hydrogen Bond Acceptor Count 14.0
Molecular Weight 833.9
Covalent Unit Count 1.0
Total Atom Stereocenter Count 12.0
Total Bond Stereocenter Count 0.0
Esol -6.637953600000002
Inchi InChI=1S/C45H55NO14/c1-9-23(2)39(52)46-33(27-16-12-10-13-17-27)34(50)41(54)58-29-21-45(55)38(59-40(53)28-18-14-11-15-19-28)36-43(8,30(49)20-31-44(36,22-56-31)60-26(5)48)37(51)35(57-25(4)47)32(24(29)3)42(45,6)7/h10-19,23,29-31,33-36,38,49-50,55H,9,20-22H2,1-8H3,(H,46,52)/t23?,29-,30-,31+,33-,34+,35+,36-,38-,43+,44-,45+/m0/s1
Smiles CCC(C)C(=O)N[C@@H](C1=CC=CC=C1)[C@H](C(=O)O[C@H]2C[C@]3([C@H]([C@H]4[C@@]([C@H](C[C@@H]5[C@]4(CO5)OC(=O)C)O)(C(=O)[C@@H](C(=C2C)C3(C)C)OC(=O)C)C)OC(=O)C6=CC=CC=C6)O)O
Nring 6.0
Defined Bond Stereocenter Count 0.0

  • 1. Outgoing r'ship FOUND_IN to/from Taxus Baccata (Plant) Rel Props:Source_db:cmaup_ingredients