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[(1R,2S,4R,5S,6R,7S,8S,10R,11R)-5-[(3aS,5S,6aS)-3a,4,5,6a-tetrahydrofuro[2,3-b]furan-5-yl]-2,10-diacetyloxy-4,5-dimethylspiro[9-oxatricyclo[6.2.2.01,6]dodecane-11,2'-oxirane]-7-yl] (E)-2-methylbut-2-enoate

PubChem CID: 102056204

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Ghose Rule False
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 119.0
Hydrogen Bond Donor Count 0.0
Pfizer 3 75 Rule False
Scaffold Graph Level C1CC2CC(C3CCCC45CCC(CC34)CC53CC3)CC2C1
Np Classifier Class Colensane and Clerodane diterpenoids
Deep Smiles C/C=C/C=O)O[C@@H][C@H]O[C@@H][C@@][C@H]6[C@@]C)[C@@H]C[C@@H][C@H]O5)OC=C5)))))))[C@H]C)C[C@@H]6OC=O)C))))))))[C@@]C6)OC3))))OC=O)C)))))))))C
Heavy Atom Count 39.0
Classyfire Class Carboxylic acids and derivatives
Scaffold Graph Node Level C1CC(C2CC3CCOC3O2)C2CC3CC4(CO4)C2(C1)CO3
Classyfire Subclass Tricarboxylic acids and derivatives
Isotope Atom Count 0.0
Molecular Complexity 1130.0
Database Name imppat_phytochem;pubchem
Defined Atom Stereocenter Count 12.0
Iupac Name [(1R,2S,4R,5S,6R,7S,8S,10R,11R)-5-[(3aS,5S,6aS)-3a,4,5,6a-tetrahydrofuro[2,3-b]furan-5-yl]-2,10-diacetyloxy-4,5-dimethylspiro[9-oxatricyclo[6.2.2.01,6]dodecane-11,2'-oxirane]-7-yl] (E)-2-methylbut-2-enoate
Veber Rule True
Classyfire Superclass Organic acids and derivatives
Xlogp 3.3
Gsk 4 400 Rule False
Molecular Formula C29H38O10
Scaffold Graph Node Bond Level C1=CC2CC(C3CCCC45COC(CC34)CC53CO3)OC2O1
Inchi Key QSTDMNRGSLDDJV-ZWDVYROGSA-N
Silicos It Class Soluble
Rotatable Bond Count 8.0
Synonyms jodrellin t
Esol Class Moderately soluble
Functional Groups C/C=C(C)C(=O)OC, CC(=O)OC, CC(=O)O[C@H](C)OC, CO[C@H]1CC=CO1, C[C@@]1(C)CO1
Compound Name [(1R,2S,4R,5S,6R,7S,8S,10R,11R)-5-[(3aS,5S,6aS)-3a,4,5,6a-tetrahydrofuro[2,3-b]furan-5-yl]-2,10-diacetyloxy-4,5-dimethylspiro[9-oxatricyclo[6.2.2.01,6]dodecane-11,2'-oxirane]-7-yl] (E)-2-methylbut-2-enoate
Exact Mass 546.246
Formal Charge 0.0
Monoisotopic Mass 546.246
Hydrogen Bond Acceptor Count 10.0
Molecular Weight 546.6
Gi Absorption True
Covalent Unit Count 1.0
Total Atom Stereocenter Count 12.0
Total Bond Stereocenter Count 1.0
Lipinski Rule Of 5 True
Inchi InChI=1S/C29H38O10/c1-7-14(2)24(32)39-22-19-12-28(13-34-28)29(26(37-19)36-17(5)31)21(35-16(4)30)10-15(3)27(6,23(22)29)20-11-18-8-9-33-25(18)38-20/h7-9,15,18-23,25-26H,10-13H2,1-6H3/b14-7+/t15-,18-,19+,20+,21+,22-,23-,25+,26+,27-,28+,29-/m1/s1
Smiles C/C=C(\C)/C(=O)O[C@@H]1[C@@H]2C[C@]3(CO3)[C@]4([C@H]1[C@@]([C@@H](C[C@@H]4OC(=O)C)C)(C)[C@@H]5C[C@H]6C=CO[C@H]6O5)[C@H](O2)OC(=O)C
Np Classifier Biosynthetic Pathway Terpenoids
Defined Bond Stereocenter Count 1.0
Egan Rule True
Np Classifier Superclass Diterpenoids