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(1R,2S,5S,6S,9S,10S,12S,13R)-16-(dimethylamino)-6,7,13-trimethyl-7-azapentacyclo[10.8.0.02,9.05,9.013,18]icos-18-en-10-ol

PubChem CID: 101672378

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Ghose Rule True
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 26.7
Hydrogen Bond Donor Count 1.0
Pfizer 3 75 Rule False
Scaffold Graph Level C1CCC2C(C1)CCC1C2CCC23CCCC2CCC13
Np Classifier Class Steroidal alkaloids
Deep Smiles CNCCC[C@]C=CC[C@@H][C@@H]6C[C@H]O)[C@@][C@H]6CC[C@@H]5[C@@H]NC8)C))C)))))))))))))C6))C)))))C
Heavy Atom Count 27.0
Classyfire Class Steroids and steroid derivatives
Scaffold Graph Node Level C1CCC2C(C1)CCC1C2CCC23CNCC2CCC13
Classyfire Subclass Steroidal alkaloids
Isotope Atom Count 0.0
Molecular Complexity 644.0
Database Name imppat_phytochem;pubchem
Defined Atom Stereocenter Count 8.0
Iupac Name (1R,2S,5S,6S,9S,10S,12S,13R)-16-(dimethylamino)-6,7,13-trimethyl-7-azapentacyclo[10.8.0.02,9.05,9.013,18]icos-18-en-10-ol
Veber Rule True
Classyfire Superclass Lipids and lipid-like molecules
Xlogp 3.7
Gsk 4 400 Rule True
Molecular Formula C24H40N2O
Scaffold Graph Node Bond Level C1=C2CCCCC2C2CCC34CNCC3CCC4C2C1
Inchi Key QESDNCVYXJTJRY-IINYINBQSA-N
Silicos It Class Soluble
Rotatable Bond Count 1.0
Synonyms pubescimine
Esol Class Moderately soluble
Functional Groups CC=C(C)C, CN(C)C, CO
Compound Name (1R,2S,5S,6S,9S,10S,12S,13R)-16-(dimethylamino)-6,7,13-trimethyl-7-azapentacyclo[10.8.0.02,9.05,9.013,18]icos-18-en-10-ol
Exact Mass 372.314
Formal Charge 0.0
Monoisotopic Mass 372.314
Hydrogen Bond Acceptor Count 3.0
Molecular Weight 372.6
Gi Absorption True
Covalent Unit Count 1.0
Total Atom Stereocenter Count 9.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 True
Inchi InChI=1S/C24H40N2O/c1-15-19-8-9-20-18-7-6-16-12-17(25(3)4)10-11-23(16,2)21(18)13-22(27)24(19,20)14-26(15)5/h6,15,17-22,27H,7-14H2,1-5H3/t15-,17?,18-,19+,20-,21-,22-,23-,24+/m0/s1
Smiles C[C@H]1[C@H]2CC[C@@H]3[C@]2(CN1C)[C@H](C[C@H]4[C@H]3CC=C5[C@@]4(CCC(C5)N(C)C)C)O
Np Classifier Biosynthetic Pathway Alkaloids, Terpenoids
Defined Bond Stereocenter Count 0.0
Egan Rule True
Np Classifier Superclass Pseudoalkaloids

  • 1. Outgoing r'ship FOUND_IN to/from Holarrhena Pubescens (Plant) Rel Props:Reference:ISBN:9780387706375; ISBN:9788185042145