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[(1S,3S,13S,14S,17S,18S,19S,20R,21S,24R,25S)-18,19,21-triacetyloxy-24,25-dihydroxy-3,13,14,25-tetramethyl-6,15,22-trioxo-2,5,16-trioxa-11-azapentacyclo[15.7.1.01,20.03,23.07,12]pentacosa-7(12),8,10-trien-20-yl]methyl acetate

PubChem CID: 101288255

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Ghose Rule False
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 237.0
Hydrogen Bond Donor Count 2.0
Pfizer 3 75 Rule True
Scaffold Graph Level CC1CCC2CCCCC2C(C)CCC2CC34CC(CCC3CC(C)C2C4)C1
Np Classifier Class Pyridine alkaloids
Deep Smiles CC=O)OC[C@][C@H]OC=O)C)))[C@H]OC=O)C)))[C@H][C@][C@]6O[C@]CC=O)[C@H]%11OC=O)C)))))[C@H]5O)))C)COC=O)cc[C@H][C@@H]C=O)O%14))C))C))nccc6))))))))))))C)O
Heavy Atom Count 51.0
Scaffold Graph Node Level OC1CCC2NCCCC2C(O)OCC2OC34CC(CCC3CC(O)C2C4)O1
Isotope Atom Count 0.0
Molecular Complexity 1500.0
Database Name imppat_phytochem;pubchem
Defined Atom Stereocenter Count 11.0
Iupac Name [(1S,3S,13S,14S,17S,18S,19S,20R,21S,24R,25S)-18,19,21-triacetyloxy-24,25-dihydroxy-3,13,14,25-tetramethyl-6,15,22-trioxo-2,5,16-trioxa-11-azapentacyclo[15.7.1.01,20.03,23.07,12]pentacosa-7(12),8,10-trien-20-yl]methyl acetate
Veber Rule False
Classyfire Superclass Alkaloids and derivatives
Xlogp -0.5
Gsk 4 400 Rule False
Molecular Formula C34H41NO16
Scaffold Graph Node Bond Level O=C1CCc2ncccc2C(=O)OCC2OC34CC(CCC3CC(=O)C2C4)O1
Inchi Key GARAEILXWIXANX-JSIPNFJXSA-N
Silicos It Class Moderately soluble
Rotatable Bond Count 9.0
Synonyms evorine
Esol Class Soluble
Functional Groups CC(=O)OC, CC(C)=O, CO, COC, COC(C)=O, cC(=O)OC, cnc
Compound Name [(1S,3S,13S,14S,17S,18S,19S,20R,21S,24R,25S)-18,19,21-triacetyloxy-24,25-dihydroxy-3,13,14,25-tetramethyl-6,15,22-trioxo-2,5,16-trioxa-11-azapentacyclo[15.7.1.01,20.03,23.07,12]pentacosa-7(12),8,10-trien-20-yl]methyl acetate
Exact Mass 719.243
Formal Charge 0.0
Monoisotopic Mass 719.243
Hydrogen Bond Acceptor Count 17.0
Molecular Weight 719.7
Gi Absorption False
Covalent Unit Count 1.0
Total Atom Stereocenter Count 12.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 False
Inchi InChI=1S/C34H41NO16/c1-14-15(2)29(42)50-27-24(47-17(4)37)28(49-19(6)39)33(13-45-16(3)36)26(48-18(5)38)23(40)21-25(41)34(33,32(27,8)44)51-31(21,7)12-46-30(43)20-10-9-11-35-22(14)20/h9-11,14-15,21,24-28,41,44H,12-13H2,1-8H3/t14-,15-,21?,24+,25+,26+,27-,28+,31+,32-,33-,34-/m0/s1
Smiles C[C@H]1[C@@H](C(=O)O[C@H]2[C@H]([C@H]([C@@]3([C@@H](C(=O)C4[C@H]([C@@]3([C@@]2(C)O)O[C@@]4(COC(=O)C5=C1N=CC=C5)C)O)OC(=O)C)COC(=O)C)OC(=O)C)OC(=O)C)C
Np Classifier Biosynthetic Pathway Alkaloids
Defined Bond Stereocenter Count 0.0
Egan Rule False
Np Classifier Superclass Nicotinic acid alkaloids

  • 1. Outgoing r'ship FOUND_IN to/from Euonymus Hamiltonianus (Plant) Rel Props:Reference:https://doi.org/10.2174/0929867033456729